SCHEMBL4043965

SCHEMBL4043965

CN(C)CCCOCc1cc2c(s1)-c1cc(Br)ccc1Sc1ccccc1-2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
HTR1A P08908 7/20 0.34
CYP1A2 P05177 7/20 0.34
CYP2D6 P10635 7/20 0.34
CHRM2 P08172 6/20 0.34
ADRA2A P08913 6/20 0.34
CHRM1 P11229 6/20 0.34
DRD1 P21728 6/20 0.34
SLC6A2 P23975 6/20 0.34
SLC6A4 P31645 6/20 0.34
OPRM1 P35372 6/20 0.34
DRD3 P35462 6/20 0.34
LMNA P02545 6/20 0.34
DRD2 P14416 5/20 0.34
ADRA1A P35348 5/20 0.34
KCNH2 Q12809 5/20 0.34
SLC6A3 Q01959 5/20 0.34
CYP2C19 P33261 5/20 0.34
HRH1 P35367 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4037158 0.99 KMT2A (0.36) KMT2AMEN1HTR1ACYP1A2CYP2D6
SCHEMBL4037482 0.94 CHRM2 (0.38) KMT2AMEN1HTR1ACYP1A2CYP2D6
SCHEMBL4040292 0.93 KMT2A (0.38) KMT2AMEN1HTR1ACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL4037222 0.93 CHRM2 (0.37) KMT2AMEN1HTR1ACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL4042137 0.92 KMT2A (0.40) KMT2AMEN1HTR1ACYP1A2CYP2D6
SCHEMBL4039594 0.90 MEN1 (0.39) KMT2AMEN1HTR1ACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL4037809 0.89 KMT2A (0.40) KMT2AMEN1HTR1ACYP1A2CYP2D6
SCHEMBL6331870 0.88 MEN1 (0.35) KMT2AMEN1HTR1ACYP1A2CYP2D6
SCHEMBL4040369 0.88 LMNA (0.48) KMT2AMEN1HTR1ACYP1A2CYP2D6
SCHEMBL4039813 0.88 MEN1 (0.35) KMT2AMEN1HTR1ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1284977-B1 THIENODIBENZOAZULENE COMPOUNDS AS TUMOR NECROSIS FACTOR INHIBITORS GLAXOSMITHKLINE ZAGREB (HR) 2009-06-24 EP claimed