SCHEMBL4040341

SCHEMBL4040341

CCCCC(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.42
KMT2A Q03164 1/20 0.41
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
PARP4 Q9UKK3 1/20 0.40
PARP3 Q9Y6F1 1/20 0.40
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
NAPRT Q6XQN6 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210597 0.90 PARP1 (0.40) PAX8TNKSPARP1PARP2PARP4
SCHEMBL4040339 0.85 TNKS (0.39) PAX8KMT2ATNKSPARP1PARP2
SCHEMBL4039947 0.83 TNKS (0.38) PAX8KMT2ATNKSPARP1PARP2
SCHEMBL6209605 0.83 DPP4 (0.44) ALDH1A1KDM4ENAMPTPOLB
SCHEMBL6208825 0.81 PAX8 (0.40) PAX8TNKSPARP1PARP2PARP4
SCHEMBL6210592 0.81 PAX8 (0.40) PAX8TNKSPARP1PARP2PARP4
SCHEMBL6212212 0.81 PTAFR (0.42) ALDH1A1POLB
SCHEMBL4047662 0.80 CTSK (0.41) PAX8TNKSPARP1PARP2PARP4
SCHEMBL5941500 0.80 NAMPT (0.46) ALDH1A1NAMPT
SCHEMBL4039942 0.79 PARP1 (0.38) PAX8TNKSPARP1PARP2PARP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed