SCHEMBL4040595

SCHEMBL4040595

CC(C)CC(CC(=O)N1CCNCC1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccc[n+]1[O-]

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.34
MC4R P32245 1/20 0.34
ALDH1A1 P00352 2/20 0.32
GAA P10253 2/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.31
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TMPRSS11D O60235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039499 0.92 CTSK (0.35) CTSKALDH1A1GAAKMT2ALMNA
SCHEMBL4039943 0.91 POLB (0.35) CTSKALDH1A1GAAKMT2ALMNA
SCHEMBL4045822 0.89 KDM4E (0.40) CTSKALDH1A1GAAKMT2APKM
SCHEMBL4040674 0.88 POLB (0.37) ALDH1A1KMT2ALMNAPKMSMN1; SMN2
SCHEMBL4043419 0.88 CTSK (0.33) CTSK
SCHEMBL4041865 0.88 ALDH1A1 (0.34) CTSKMC4RALDH1A1GAAKMT2A
SCHEMBL4040117 0.86 CTSK (0.32) CTSK
SCHEMBL4044086 0.83 CTSK (0.40) CTSK
SCHEMBL4041828 0.82 CTSK (0.35) CTSKMC4RALDH1A1GAAKMT2A
SCHEMBL6211805 0.81 CTSK (0.35) CTSKMC4RALDH1A1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1463728-B1 FUSED CYCLIC MODULATORS OF NUCLEAR HORMONE RECEPTOR FUNCTION BRISTOL MYERS SQUIBB CO (US) 2009-01-14 EP disclosed