SCHEMBL4041214

SCHEMBL4041214

Nc1nccnc1NC(=O)C1CN(C(=O)O)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 1/20 0.38
ATR Q13535 1/20 0.34
MAP4K4 O95819 1/20 0.34
GSK3B P49841 4/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
JAK2 O60674 3/20 0.32
TYK2 P29597 3/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13905150 0.81 GSK3B (0.46) GSK3BTSHRJAK2TYK2
SCHEMBL4045594 0.80 PTPN2 (0.44) HDAC1HDAC2NPC1RAB9A
SCHEMBL19597568 0.71 ATR (0.44) NEK2ATRALDH1A1NPC1RAB9A
SCHEMBL5494591 0.68 HDAC3 (0.36) TSHRALDH1A1PIM1PIM3PIM2
SCHEMBL29085989 0.67 DEGS1 (0.60) NPC1RAB9A
SCHEMBL29200836 0.67 L3MBTL1 (0.41) ATRALDH1A1
SCHEMBL15797955 0.66 CA12 (0.33) ALDH1A1
SCHEMBL2590028 0.65 HDAC2 (0.51) TSHRHDAC3HDAC1HDAC2
SCHEMBL18138923 0.65 GSK3B (0.39) GSK3BHDAC3HDAC1HDAC2
SCHEMBL2595612 0.65 GAA (0.50) TSHRHDAC3HDAC1HDAC2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed
WO-2009016046-A2 SUNLESS TANNING COMPOSITIONS COMPRISING SUBSTITUTED POLYAMINE COMPOUNDS BASF SE (CH) 2009-02-05 WO disclosed