SCHEMBL4041327

SCHEMBL4041327

C[C@@H](CN1CCOCC1)N(OC(C)(C)C)C(=O)CCC(NC(=O)OC(C)(C)C)C1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
CTSK P43235 5/20 0.35
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CTSL P07711 3/20 0.33
CTSB P07858 3/20 0.33
ITGB3 P05106 8/20 0.32
ITGA2B P08514 8/20 0.32
CTSS P25774 2/20 0.32
CTSD P07339 1/20 0.32
TACR2 P21452 1/20 0.31
TACR3 P29371 1/20 0.31
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1414479 1.00 ALDH1A1 (0.35) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL30968576 0.82 CTSK (0.42) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL1414550 0.78 MEN1 (0.37) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL1414548 0.78 MEN1 (0.37) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL1414546 0.78 MEN1 (0.37) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL13821640 0.73 EPHX1 (0.44) CTSKHDAC4HDAC1HDAC6CTSL
SCHEMBL2813531 0.72 HDAC4 (0.42) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL2813537 0.72 HDAC4 (0.42) ALDH1A1CTSKHDAC4HDAC1HDAC6
SCHEMBL1414317 0.71 HDAC4 (0.46) CTSKHDAC4HDAC1HDAC6ITGB3
SCHEMBL1414320 0.71 HDAC4 (0.46) CTSKHDAC4HDAC1HDAC6ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531545-B2 2-amino-3,4-dihydro-pyrido[3,4-d]pyrimidine derivatives useful as inhibitors of β-secretase (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2009-05-12 US disclosed
US-20070259898-A1 NOVEL 2-AMINO-3,4-DIHYDRO-PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF beta-SECRETASE (BACE) BAXTER ELLEN E 2007-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070259898-A1 NOVEL 2-AMINO-3,4-DIHYDRO-PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF beta-SECRETASE (BACE) BACE2, PSEN2, BACE1 ALDH1A1 3796/4885CTSK 1040/4885HDAC4 3098/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.