SCHEMBL4041610

SCHEMBL4041610

COc1ccc2cc(CCC3(O)CCC(NCc4ccc5c(n4)NC(=O)CO5)CC3)ccc2n1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 19/20 0.54
KCNQ1 P51787 1/20 0.48
CACNA1C Q13936 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044878 0.85 KCNH2 (0.47) KCNH2
SCHEMBL5261640 0.84 KCNH2 (0.67) KCNH2
SCHEMBL14498893 0.84 KCNH2 (0.67) KCNH2
SCHEMBL13407407 0.84 KCNH2 (0.54) KCNH2
SCHEMBL3582737 0.84 KCNH2 (0.54) KCNH2
SCHEMBL4507055 0.84 KCNH2 (0.54) KCNH2
SCHEMBL14524460 0.80 KCNH2 (0.60) KCNH2KCNQ1CACNA1C
SCHEMBL14498851 0.77 KCNH2 (0.69) KCNH2
SCHEMBL5651296 0.76 KCNH2 (0.56) KCNH2
SCHEMBL5653812 0.76 KCNH2 (0.56) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537123-B1 AMINO-SUBSTITUTED CYCLOHEXANE DERIVATIVES FOR THE TREATMENT OF BACTERIAL INFECTIONS GLAXO GROUP LTD (GB) 2009-04-29 EP claimed