SCHEMBL4042729

SCHEMBL4042729

Cc1cccc(C2(C(C(=O)NC3CCCCC3)C3CCCCC3)Nc3ccccc3N2)c1C

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
EPHX1 P07099 1/20 0.43
GAA P10253 2/20 0.41
ALOX12 P18054 2/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
TSHR P16473 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043366 0.89 TSHR (0.50) HPGDRAB9ANPC1KMT2AMEN1
SCHEMBL4036690 0.84 TSHR (0.43) HPGDRAB9ANPC1GAALMNA
SCHEMBL4039455 0.84 KMT2A (0.48) HPGDRAB9ANPC1LMNAKMT2A
SCHEMBL4041189 0.84 NPC1 (0.41) HPGDRAB9ANPC1LMNAKMT2A
SCHEMBL4039913 0.84 TSHR (0.46) HPGDRAB9ANPC1EPHX1LMNA
SCHEMBL4044888 0.83 KMT2A (0.45) RAB9ANPC1KMT2AMEN1TSHR
SCHEMBL4044962 0.83 KMT2A (0.49) HPGDEPHX1KMT2AMEN1TSHR
SCHEMBL4044367 0.83 PKM (0.40) HPGDRAB9ANPC1EPHX1LMNA
SCHEMBL4044346 0.82 EPHX1 (0.47) HPGDRAB9ANPC1EPHX1KMT2A
SCHEMBL4037704 0.82 TSHR (0.41) HPGDRAB9ANPC1EPHX1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038259-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F.HOFFMANN-LA ROCHE AG (CH) 2009-03-25 EP disclosed
WO-2008000643-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F. HOFFMANN-LA ROCHE AG (CH) 2008-01-03 WO disclosed