SCHEMBL4044962

SCHEMBL4044962

CCc1ccccc1C1(C(C(=O)NC2CCCCC2)C2CCCCC2)Nc2ccccc2N1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
TSHR P16473 4/20 0.42
HSD17B10 Q99714 2/20 0.42
HTT P42858 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MEN1 O00255 2/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
TP53 P04637 2/20 0.38
C3AR1 Q16581 1/20 0.38
EPHX1 P07099 1/20 0.38
HPGD P15428 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036690 0.85 TSHR (0.43) KMT2ATSHRHSD17B10HTTKDM4E
SCHEMBL4044158 0.85 GAA (0.47) KMT2ATSHRHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL4039455 0.85 KMT2A (0.48) KMT2ATSHRHSD17B10HTTKDM4E
SCHEMBL4044367 0.83 PKM (0.40) KMT2ATSHRHSD17B10HTTKDM4E
SCHEMBL4042729 0.83 HPGD (0.44) KMT2ATSHRHTTALDH1A1SMN1; SMN2
SCHEMBL4044939 0.83 NPC1 (0.46) KMT2ATSHRHSD17B10HTTKDM4E
SCHEMBL4044888 0.82 KMT2A (0.45) KMT2ATSHRHSD17B10HTTKDM4E
SCHEMBL4039869 0.82 HPGD (0.45) KMT2ATSHRALDH1A1MEN1HPGD
SCHEMBL4043366 0.82 TSHR (0.50) KMT2ATSHRHSD17B10HTTKDM4E
SCHEMBL4042940 0.81 TSHR (0.45) KMT2ATSHRHSD17B10HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038259-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F.HOFFMANN-LA ROCHE AG (CH) 2009-03-25 EP disclosed
WO-2008000643-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F. HOFFMANN-LA ROCHE AG (CH) 2008-01-03 WO disclosed