SCHEMBL4044482

SCHEMBL4044482

Cc1ccoc1C1(C(C(=O)NC2CCCCC2)C2CCCCC2)Nc2ccccc2N1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
GLA P06280 1/20 0.44
MAPK1 P28482 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HPGD P15428 4/20 0.41
POLB P06746 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 3/20 0.39
GAA P10253 2/20 0.39
TSHR P16473 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034516 0.81 HPGD (0.45) HPGDPOLBNPSR1MEN1KMT2A
SCHEMBL4039067 0.80 NPC1 (0.44) NPC1RAB9AHPGDPOLBMEN1
SCHEMBL4042729 0.80 HPGD (0.44) LMNANPC1RAB9AHPGDMEN1
SCHEMBL4042940 0.79 TSHR (0.45) LMNANPC1RAB9AHPGDPOLB
SCHEMBL4036317 0.79 HPGD (0.43) NPC1RAB9AHPGDPOLBMEN1
SCHEMBL4044722 0.79 RAB9A (0.41) NPC1RAB9AHPGDMEN1KMT2A
SCHEMBL4039913 0.79 TSHR (0.46) LMNANPC1RAB9AHPGDMEN1
SCHEMBL4041189 0.79 NPC1 (0.41) LMNANPC1RAB9AHPGDMEN1
SCHEMBL4038863 0.78 GAA (0.39) NPC1RAB9AHPGDPOLBNPSR1
SCHEMBL4044713 0.78 KMT2A (0.44) LMNANPC1RAB9AHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038259-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F.HOFFMANN-LA ROCHE AG (CH) 2009-03-25 EP disclosed
WO-2008000643-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F. HOFFMANN-LA ROCHE AG (CH) 2008-01-03 WO disclosed