SCHEMBL4044807

SCHEMBL4044807

CC(C)CC(NC(=O)Oc1ccco1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.39
CTSL P07711 6/20 0.38
CTSS P25774 5/20 0.38
SMYD3 Q9H7B4 2/20 0.36
CTSB P07858 2/20 0.35
ALDH1A1 P00352 1/20 0.34
FKBP1A P62942 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051063 0.92 SMYD3 (0.36) CTSKCTSLCTSSSMYD3ALDH1A1
SCHEMBL4049641 0.89 CTSK (0.40) CTSKCTSLCTSSSMYD3CTSB
SCHEMBL4048306 0.88 CTSK (0.38) CTSKCTSLCTSSSMYD3CTSB
SCHEMBL4047069 0.88 CTSK (0.42) CTSKCTSLCTSSCTSB
SCHEMBL4040754 0.87 CTSK (0.40) CTSKCTSLCTSSCTSB
SCHEMBL4050718 0.87 CTSK (0.41) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4043952 0.87 CTSK (0.42) CTSKCTSLCTSSCTSBFKBP1A
SCHEMBL4043196 0.87 CTSK (0.39) CTSKCTSLCTSSSMYD3CTSB
SCHEMBL4044450 0.86 CTSK (0.43) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4042866 0.86 CTSK (0.50) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed