SCHEMBL4044993

SCHEMBL4044993

CCc1cc(C(=O)O)c([N+](=O)[O-])c(OC)c1OCCCN1CCOCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
ALDH1A1 P00352 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
CYP2D6 P10635 3/20 0.47
TSHR P16473 1/20 0.47
PKM P14618 1/20 0.47
CYP1A2 P05177 2/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 3/20 0.43
POLB P06746 1/20 0.43
SYK P43405 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTR1A P08908 1/20 0.41
CYP3A4 P08684 1/20 0.41
HRH3 Q9Y5N1 2/20 0.41
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043734 0.85 CYP2D6 (0.48) KDM4EALDH1A1CYP2D6TSHRCYP1A2
SCHEMBL6437918 0.85 KDM4E (0.52) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL7718548 0.85 CYP2D6 (0.50) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL31620997 0.84 KDM4E (0.58) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL31620995 0.76 KDM4E (0.54) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL31621003 0.76 KDM4E (0.54) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL4044992 0.76 ALDH1A1 (0.54) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL7526518 0.76 KDM4E (0.64) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL5567501 0.76 KDM4E (0.64) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A
SCHEMBL4047895 0.73 KDM4E (0.53) KDM4ESMN1; SMN2ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103719-A1 SUBSTITUTED 4-(INDOL-3-YL)QUINAZOLINES AND USE AND PRODUCTION THEREOF FREIE UNIVERSITÄT BERLIN (DE) 2009-08-27 WO disclosed