SCHEMBL4043734

SCHEMBL4043734

CCc1cc(C(=O)O)c(N)c(OC)c1OCCCN1CCOCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.48
TSHR P16473 1/20 0.48
POLB P06746 1/20 0.46
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 2/20 0.43
HRH3 Q9Y5N1 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
HTR2A P28223 1/20 0.43
SCN1A P35498 1/20 0.43
HTR2B P41595 1/20 0.43
KCNH2 Q12809 1/20 0.43
SCN2A Q99250 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
SCN3A Q9NY46 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044993 0.85 KDM4E (0.49) CYP2D6TSHRPOLBLMNAKDM4E
SCHEMBL7718571 0.84 CYP2D6 (0.51) CYP2D6TSHRPOLBLMNAKDM4E
SCHEMBL6442664 0.84 KDM4E (0.47) CYP2D6TSHRPOLBLMNAKDM4E
SCHEMBL11642461 0.77 KDM4E (0.46) POLBKDM4ETDP1ALDH1A1MEN1
SCHEMBL6447784 0.76 TSHR (0.60) CYP2D6TSHRPOLBLMNAKDM4E
SCHEMBL4047895 0.76 KDM4E (0.53) CYP2D6TSHRPOLBLMNAKDM4E
SCHEMBL4043732 0.74 ALDH1A1 (0.48) CYP2D6TSHRPOLBKDM4ETDP1
SCHEMBL7718548 0.73 CYP2D6 (0.50) CYP2D6TSHRPOLBLMNAKDM4E
SCHEMBL6437918 0.73 KDM4E (0.52) CYP2D6TSHRLMNAKDM4ETDP1
SCHEMBL28824456 0.72 CYP2D6 (0.49) CYP2D6TSHRLMNAKDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103719-A1 SUBSTITUTED 4-(INDOL-3-YL)QUINAZOLINES AND USE AND PRODUCTION THEREOF FREIE UNIVERSITÄT BERLIN (DE) 2009-08-27 WO disclosed