SCHEMBL4045501

SCHEMBL4045501

CC(C)COC(=O)ON1CC(=O)C2C1CCN2C(=O)C(CC(C)C)NC(=O)c1ccc(-c2cccs2)cc1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 17/20 0.53
CTSS P25774 5/20 0.41
HPGDS O60760 1/20 0.40
CTSL P07711 3/20 0.40
CTSB P07858 2/20 0.40
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046409 0.90 CTSK (0.57) CTSKCTSSHPGDSCTSLCTSB
SCHEMBL4044462 0.90 CTSK (0.54) CTSKCTSSHPGDSCTSLCTSB
SCHEMBL4046312 0.89 CTSK (0.52) CTSKCTSSHPGDSCTSLCTSB
SCHEMBL4041020 0.87 CTSK (0.54) CTSKCTSSHPGDSCTSLCTSB
SCHEMBL4043121 0.87 CTSK (0.56) CTSKCTSSCTSL
SCHEMBL4050211 0.86 CTSK (0.69) CTSKCTSSCTSL
SCHEMBL4042616 0.86 CTSK (0.59) CTSKCTSSHPGDSCTSLCTSB
SCHEMBL4041651 0.85 CTSK (0.55) CTSKCTSSCTSL
SCHEMBL4045325 0.85 CTSK (0.69) CTSKCTSSCTSLCTSB
SCHEMBL4043531 0.85 CTSK (0.62) CTSKCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed