SCHEMBL4045677

SCHEMBL4045677

CC(C[CH]C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccncc1)C(N)=O

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.34
SMYD3 Q9H7B4 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049235 0.91 TSHR (0.38) HSD11B1
SCHEMBL4039217 0.89 HSD17B10 (0.40) SMYD3
SCHEMBL4044364 0.87 AKR1C3 (0.31)
SCHEMBL4037609 0.85 CTSK (0.31)
SCHEMBL4041823 0.85 CTSK (0.39)
SCHEMBL4044693 0.84 CTSK (0.42)
SCHEMBL4040282 0.82 PIK3CD (0.35)
SCHEMBL4044949 0.82 SMYD3 (0.38) SMYD3
SCHEMBL4044726 0.81 PARP1 (0.34)
SCHEMBL4039452 0.81 CTSK (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed