SCHEMBL4045684

SCHEMBL4045684

CC(=O)c1ccc(C2CCCCN2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C19 P33261 2/20 0.45
CHRNB2 P17787 2/20 0.45
CHRNA7 P36544 2/20 0.45
CHRNA4 P43681 2/20 0.45
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2A6 P11509 1/20 0.45
CYP2C9 P11712 1/20 0.45
PARP1 P09874 3/20 0.43
PARP2 Q9UGN5 2/20 0.43
MKNK1 Q9BUB5 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
EPHX1 P07099 1/20 0.41
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21806659 0.95 MKNK1 (0.46) MEN1KMT2ACYP2D6CYP2C19CHRNB2
SCHEMBL16401323 0.85 KMT2A (0.46) MEN1KMT2ACYP2D6CYP2C19CHRNB2
SCHEMBL4045246 0.85 KMT2A (0.46) MEN1KMT2ACYP2D6CYP2C19CHRNB2
SCHEMBL26693436 0.83 PARP1 (0.51) MEN1KMT2ACYP2D6CYP2C19CHRNB2
SCHEMBL3529098 0.83 ALDH1A1 (0.47) MEN1KMT2ACYP2D6CYP2C19POLB
SCHEMBL17782257 0.83 ALDH1A1 (0.47) MEN1KMT2ACYP2D6CYP2C19POLB
SCHEMBL4767634 0.82 PARP1 (0.50) MEN1KMT2ACYP2D6CYP2C19CHRNB2
Hydrochloric Acid SCHEMBL17782206 0.81 ALDH1A1 (0.46) MEN1KMT2ACYP2D6CYP2C19SMN1; SMN2
Hydrochloric Acid SCHEMBL1652940 0.81 ALDH1A1 (0.46) MEN1KMT2ACYP2D6CYP2C19SMN1; SMN2
Acetic Acid SCHEMBL28115056 0.81 MEN1 (0.54) MEN1KMT2ACYP2D6CYP2C19CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103478-A1 PYRIDONE AND PYRIDAZINONE DERIVATIVES AS MCH ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-08-27 WO disclosed