SCHEMBL4046402

SCHEMBL4046402

COc1cc(C(=O)N(C)OC)ccc1CO

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
BLM P54132 1/20 0.46
ELANE P08246 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MLYCD O95822 1/20 0.42
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13664923 0.80 CYP1A2 (0.45) CYP1A2HSP90AA1HSP90AB1BLMELANE
SCHEMBL4050727 0.79 PKM (0.56) CYP1A2MEN1KMT2AALDH1A1PDCD1
SCHEMBL2424457 0.79 CA12 (0.65) TSHRCA12CA1CA2CA4
SCHEMBL17894222 0.79 MLYCD (0.42) CYP1A2HSP90AA1HSP90AB1BLMMEN1
SCHEMBL4568348 0.78 MLYCD (0.48) CYP1A2HSP90AA1HSP90AB1BLMELANE
SCHEMBL5604944 0.78 CYP1A2 (0.44) CYP1A2HSP90AA1HSP90AB1BLMELANE
SCHEMBL4181181 0.78 MAPK1 (0.60) ELANEALDH1A1TSHRPDE4APDE4B
SCHEMBL13451040 0.78 MAPK1 (0.59) CYP1A2MEN1KMT2AALDH1A1PDCD1
SCHEMBL2252810 0.78 MAPT (0.58) CYP1A2MEN1KMT2AALDH1A1PDCD1
SCHEMBL1014530 0.77 MAPT (0.51) MEN1KMT2AALDH1A1CYP2C9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103478-A1 PYRIDONE AND PYRIDAZINONE DERIVATIVES AS MCH ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-08-27 WO disclosed