SCHEMBL4048369

SCHEMBL4048369

CN(C)C1(Cc2cccc(Cl)c2)CCC(C(N)=O)CC1.CN(C)C1(Cc2ccccc2F)CCC(NC(=O)CCC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
SIGMAR1 Q99720 6/20 0.40
ACKR3 P25106 3/20 0.37
KMT2A Q03164 4/20 0.36
HPGD P15428 2/20 0.36
THRB P10828 1/20 0.36
EPHX2 P34913 1/20 0.35
MEN1 O00255 3/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPK1 P28482 1/20 0.34
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048372 0.93 NPC1 (0.42) NPC1SIGMAR1ACKR3KMT2AHPGD
SCHEMBL4048483 0.89 SIGMAR1 (0.48) NPC1SIGMAR1ACKR3KMT2AHPGD
SCHEMBL4055346 0.85 ACKR3 (0.48) SIGMAR1ACKR3KMT2AHPGDMEN1
SCHEMBL4216689 0.84 SIGMAR1 (0.39) SIGMAR1ACKR3KMT2AMEN1ALDH1A1
SCHEMBL4052294 0.81 ACKR3 (0.48) NPC1SIGMAR1ACKR3KMT2AMEN1
SCHEMBL16143480 0.80 SIGMAR1 (0.42) SIGMAR1ACKR3KMT2AHPGDTHRB
SCHEMBL207325 0.80 NPC1 (0.49) NPC1SIGMAR1ACKR3KMT2AHPGD
SCHEMBL4054730 0.80 ACKR3 (0.50) SIGMAR1ACKR3KMT2AMEN1ALDH1A1
SCHEMBL16143615 0.78 ACKR3 (0.48) ACKR3KMT2AMEN1ALDH1A1DRD2
SCHEMBL4045470 0.78 ACKR3 (0.48) ACKR3KMT2AMEN1ALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751088-B1 OXO-SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2014-10-08 EP claimed
US-7476763-B2 Oxo-substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2009-01-13 US claimed
US-20070088034-A1 Oxo-substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-04-19 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070088034-A1 Oxo-substituted cyclohexyl-1,4-diamine compounds AOC1, ODC1, OTC NPC1 20/4885SIGMAR1 1889/4885ACKR3 3574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.