SCHEMBL4048461

SCHEMBL4048461

COc1cccc(-c2c(-c3ccncc3)nn3c4c(cnc23)CC2(CC4)OCCO2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 10/20 0.49
KDR P35968 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
LMNA P02545 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HTT P42858 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
CASP1 P29466 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052299 0.89 BRAF (0.40) BRAFKDRALDH1A1KDM4EMAPT
SCHEMBL4048686 0.87 BRAF (0.39) BRAFALDH1A1HPGDHTTMEN1
SCHEMBL4052889 0.87 BRAF (0.47) BRAFMAPK14MAPK13RAF1MAPK12
SCHEMBL4047106 0.85 BRAF (0.51) BRAFKDRMAPTTDP1MAPK14
SCHEMBL4045295 0.82 BRAF (0.46) BRAFKDRALDH1A1KDM4EMAPT
SCHEMBL4054055 0.82 BRAF (0.49) BRAFKDRALDH1A1KDM4EMAPT
SCHEMBL4047970 0.77
SCHEMBL4046191 0.75 NPC1 (0.53) BRAFKDRALDH1A1MAPTLMNA
SCHEMBL4055203 0.74 BRAF (0.46) BRAFKDRALDH1A1MAPTTDP1
SCHEMBL4054162 0.72 BRAF (0.49) BRAFMAPK14MAPK13RAF1MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108827-A1 FUSED TRICYCLIC PYRAZOLO[1, 5-A]PYRIMIDINES, METHODS FOR PREPARATION AND USES THEREOF WYETH (US) 2009-09-03 WO claimed