SCHEMBL4048972

SCHEMBL4048972

CC1(C)CCc2c(-c3ccco3)nc3sc4c(=O)[nH]cnc4c3c2C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.56
PDE4B Q07343 2/20 0.56
PDE4D Q08499 2/20 0.56
KDM4E B2RXH2 11/20 0.52
ALDH1A1 P00352 8/20 0.47
HPGD P15428 7/20 0.47
HIF1A Q16665 1/20 0.47
TDP1 Q9NUW8 3/20 0.47
HKDC1 Q2TB90 1/20 0.47
KMT2A Q03164 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
POLB P06746 4/20 0.47
CYP2C9 P11712 1/20 0.47
ADRB2 P07550 5/20 0.45
MAPT P10636 3/20 0.44
MEN1 O00255 2/20 0.44
MCL1 Q07820 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
PKM P14618 1/20 0.44
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047943 0.84 PDE4A (0.56) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4052788 0.81 PDE4B (0.64) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4045649 0.80 KDM4E (0.55) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4044859 0.77 ALDH1A1 (0.74) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4046467 0.76 KDM4E (0.61) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4046040 0.76 HPGD (0.74) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL5245426 0.75 KDM4E (0.61) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4047007 0.74 PDE4B (0.70) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4047111 0.74 KDM4E (0.60) PDE4APDE4BPDE4DKDM4EALDH1A1
SCHEMBL4047590 0.74 PDE4B (0.69) PDE4APDE4BPDE4DKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1819710-B1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES ALMIRALL LAB (ES) 2009-03-11 EP disclosed
EP-1819710-A1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES Laboratorios Almirall, S.A. (ES) 2007-08-22 EP disclosed
WO-2006058724-A1 NEW PYRIDOTHIENOPYRIMIDINE DERIVATIVES LABORATORIOS ALMIRALL, S.A. (ES) 2006-06-08 WO disclosed