SCHEMBL4051328

SCHEMBL4051328

Cc1cc(Br)ccc1-c1ncc(Br)s1.Cc1cc(Br)ccc1-c1nccs1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.36
SNCA P37840 1/20 0.35
ABL1 P00519 1/20 0.32
BCR P11274 1/20 0.32
CYP2A6 P11509 2/20 0.32
PDPK1 O15530 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
NPC1 O15118 1/20 0.32
PKM P14618 1/20 0.32
RECQL P46063 1/20 0.32
RAB9A P51151 1/20 0.32
POLB P06746 1/20 0.32
SRC P12931 2/20 0.31
SYK P43405 2/20 0.31
CHEK2 O96017 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047151 0.89 PDPK1 (0.39) CYP17A1ABL1BCRCYP2A6PDPK1
SCHEMBL4509373 0.89 SNCA (0.42) SNCAKDM4EMEN1LMNAMAPT
SCHEMBL25403240 0.76 SNCA (0.42) CYP17A1SNCAKDM4EMEN1LMNA
SCHEMBL20641436 0.74 SNCA (0.41) SNCAKDM4EMEN1LMNAMAPT
SCHEMBL11440352 0.73 ADORA2A (0.41) ABL1BCRCYP2A6PDPK1CHEK2
SCHEMBL13393593 0.73 SRC (0.47) CYP17A1PDPK1LMNAMAPTNPC1
SCHEMBL20645325 0.71 SNCA (0.39) SNCAKDM4EMEN1LMNAMAPT
SCHEMBL25405292 0.70 HSD17B1 (0.41) SNCACYP2A6KDM4EMEN1LMNA
SCHEMBL25400693 0.70 ALDH1A3 (0.38) SNCACYP2A6KDM4EMEN1LMNA
SCHEMBL25402313 0.70 SNCA (0.41) SNCAABL1KDM4EMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697333-A4 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-1697333-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS Merck & Co., Inc. (US) 2006-09-06 EP disclosed
WO-2005058848-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO., INC. (US) 2005-06-30 WO disclosed