SCHEMBL4051674

SCHEMBL4051674

O=S(=O)(C1CCN(Cc2ccccc2)CC1)n1ccc2c3nc(Cl)nc(N4CCOCC4)c3ccc21

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.47
MTOR P42345 15/20 0.41
PIK3CA P42336 14/20 0.41
ACHE P22303 1/20 0.39
HTR2A P28223 1/20 0.39
PIK3CG P48736 2/20 0.39
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049748 0.86 MAPT (0.45) HRH3MTOR
SCHEMBL4050241 0.81 HTR6 (0.47) HRH3MTORPIK3CAHTR2AHTR6
SCHEMBL4057700 0.79 HRH3 (0.58) HRH3PIK3CAPIK3CGHTR6
SCHEMBL4056388 0.78 MTOR (0.60) HRH3MTORPIK3CAHTR6
SCHEMBL4051355 0.72 PIK3CA (0.46) MTORPIK3CAPIK3CG
SCHEMBL4051692 0.71 HRH3 (0.43) HRH3MTORPIK3CA
SCHEMBL4057900 0.71 SMN1; SMN2 (0.45) HRH3MTOR
SCHEMBL4057172 0.69 MTOR (0.79) MTORPIK3CAPIK3CG
SCHEMBL3985904 0.69 PIK3CA (0.74) MTORPIK3CAPIK3CG
SCHEMBL18025696 0.69 PIK3CA (0.45) HRH3MTORPIK3CAACHEPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111547-A1 7H-PYRROLO[2,3-H]QUINAZOLINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESIS WYETH (US) 2009-09-11 WO disclosed