SCHEMBL4052669

SCHEMBL4052669

COc1ccc(CO)c2c3cc(F)ccc3n(C)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HPGD P15428 2/20 0.38
CYP19A1 P11511 2/20 0.38
NQO2 P16083 2/20 0.38
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
CASP1 P29466 1/20 0.37
HTT P42858 1/20 0.37
CASP7 P55210 1/20 0.37
ATM Q13315 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PLA2G4A P47712 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
TRPC5 Q9UL62 1/20 0.36
TSHR P16473 1/20 0.36
THRB P10828 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13693825 0.87 KDM4E (0.43) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL4053668 0.84 KDM4E (0.39) KDM4EALDH1A1HPGDCYP19A1NQO2
SCHEMBL4055213 0.81 MAPT (0.48) ALDH1A1MEN1KMT2AHPGDHTT
SCHEMBL13693826 0.76 ALDH1A1 (0.49) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL4373659 0.76 CYP19A1 (0.53) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL2908313 0.73 PDE4A (0.50) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL696497 0.71 PDCD1 (0.50) KDM4EALDH1A1KMT2AGAAHTT
SCHEMBL31280042 0.71 PDCD1 (0.50) KDM4EALDH1A1KMT2AGAAHTT
SCHEMBL4055500 0.71 KDM4E (0.39) KDM4EALDH1A1HPGDCYP19A1NQO2
SCHEMBL4541903 0.68 MYLK (0.40) KDM4EALDH1A1HPGDHTTRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed