SCHEMBL4053077

SCHEMBL4053077

CC(C)(C)C1=NCCC(c2ccc(Cl)cc2C#N)=C1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 11/20 0.33
NOS2 P35228 11/20 0.33
NOS3 P29474 10/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTAFR P25105 2/20 0.33
CNR1 P21554 4/20 0.32
CNR2 P34972 4/20 0.32
CRHR1 P34998 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17224432 0.72 MAPK10 (0.38)
Hydrochloric Acid SCHEMBL4049403 0.70 KDM4E (0.33) NOS1NOS2NOS3KDM4EMAPT
SCHEMBL17224458 0.68 AR (0.40)
SCHEMBL17224438 0.68 HTR1A (0.32)
SCHEMBL28517116 0.66 SLC6A4 (0.55)
SCHEMBL12483460 0.65 KDM4E (0.47) KDM4EMAPTTDP1CNR1CNR2
SCHEMBL19169604 0.65 AR (0.41) KDM4EMAPTTDP1
SCHEMBL4049394 0.64 HTR2C (0.55) MAPT
SCHEMBL14013151 0.63 SLC6A4 (0.40) NOS1NOS2NOS3KDM4ECNR1
SCHEMBL13525469 0.62 AR (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013214-A2 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2009-01-14 EP disclosed
WO-2007131020-A2 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-15 WO disclosed