SCHEMBL14013151

SCHEMBL14013151

N#Cc1cc(Cl)ccc1C1=CCN(Cl)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.40
DRD2 P14416 3/20 0.35
DRD4 P21917 1/20 0.35
CYP2A6 P11509 1/20 0.35
HTR6 P50406 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCNB1 P14635 1/20 0.33
CCND1 P24385 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
DRD1 P21728 1/20 0.33
AOC3 Q16853 1/20 0.32
NOS3 P29474 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28517116 0.86 SLC6A4 (0.55) SLC6A4DRD2DRD4HTR6CCNB2
SCHEMBL28510941 0.80 CNR1 (0.40) SLC6A4DRD2DRD4CNR1CCNB2
SCHEMBL27773025 0.78 KMT2A (0.41) SLC6A4DRD2DRD4HTR6OPRM1
SCHEMBL4224923 0.74 CNR1 (0.52) HTR6CNR1
SCHEMBL4049394 0.72 HTR2C (0.55) HTR6
Hydrochloric Acid SCHEMBL4049403 0.70 KDM4E (0.33) CYP2A6CNR1CNR2NOS3NOS1
SCHEMBL23551386 0.69 SLC6A4 (0.49) SLC6A4HTR6KDM4E
SCHEMBL28508682 0.67 SLC6A4 (0.57) SLC6A4DRD2DRD1NOS2
SCHEMBL1197731 0.65 AR (0.57) CNR1CNR2KDM4E
SCHEMBL8561261 0.64 XDH (0.47) CNR1CNR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470680-B2 Constrained compounds as CGRP-receptor antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-30 US disclosed
US-20070259851-A1 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY 2007-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070259851-A1 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS CALCR, BDKRB2, CALCRL SLC6A4 2592/4885DRD2 1322/4885DRD4 4004/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.