SCHEMBL4053934

SCHEMBL4053934

O=c1cc(-c2ccc(Cl)cc2)nc[nH]1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.53
PARP1 P09874 1/20 0.46
KDM5B Q9UGL1 1/20 0.45
KMO O15229 1/20 0.44
MAP4K4 O95819 3/20 0.43
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
TSHR P16473 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NOTUM Q6P988 2/20 0.41
MAPK1 P28482 1/20 0.40
CA12 O43570 1/20 0.40
ALPL P05186 1/20 0.40
METAP2 P50579 1/20 0.39
MAPKAPK2 P49137 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451431 0.81 XDH (0.49) KDM5BKMOALDH1A1KDM4EMAPT
SCHEMBL4709224 0.79 GSK3B (0.50) KDM5BMAP4K4ALDH1A1KDM4EMAPT
Hydrochloric Acid SCHEMBL29856925 0.79 XDH (0.47) KDM5BKMOALDH1A1KDM4EMAPT
SCHEMBL29417027 0.79 PARP1 (0.44) HSD11B1PARP1MAP4K4ALDH1A1
SCHEMBL4058328 0.77 PDE2A (0.47) PARP1NOTUMMAPKAPK2
SCHEMBL30952085 0.77 ABL1 (0.39) HSD11B1PARP1KDM5B
SCHEMBL21359186 0.75 KDM5B (0.39) HSD11B1KDM5BALDH1A1KDM4EMAPKAPK2
SCHEMBL10688603 0.73 PDE4A (0.59) ALDH1A1KDM4EGAAMAPTTHRB
SCHEMBL29465046 0.72 AURKA (0.40) HSD11B1PARP1KDM5BMAP4K4MAPK1
SCHEMBL16983733 0.72 PARP1 (0.41) HSD11B1PARP1KMOALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137270-A2 AZETIDINE DERIVATIVES H. LUNDBECK A/S (DK) 2009-11-12 WO disclosed
WO-2009120655-A1 INDOLE DERIVATIVES H. LUNDBECK A/S (DK) 2009-10-01 WO disclosed