SCHEMBL16983733

SCHEMBL16983733

O=c1cc(-c2cc(Cl)ccc2C(F)(F)F)nc[nH]1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.41
HCAR1 Q9BXC0 1/20 0.40
JAK2 O60674 1/20 0.39
ALDH1A1 P00352 2/20 0.38
PTGES O14684 1/20 0.36
TMPRSS4 Q9NRS4 1/20 0.36
SLC40A1 Q9NP59 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PDE2A O00408 1/20 0.35
PTP4A3 O75365 1/20 0.34
HSD11B1 P28845 2/20 0.34
CDK1 P06493 1/20 0.34
PPOX P50336 1/20 0.33
PLAT P00750 1/20 0.33
KMO O15229 1/20 0.33
STK10 O94804 1/20 0.33
SLK Q9H2G2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31252407 0.75 F11 (0.44)
SCHEMBL16115041 0.74 F11 (0.39) HCAR1ALDH1A1TMPRSS4MEN1KMT2A
SCHEMBL16974663 0.74 KMO (0.43) JAK2TMPRSS4HSD11B1KMO
SCHEMBL30561145 0.73 PARP1 (0.40) PARP1ALDH1A1HSD11B1
SCHEMBL29076917 0.73 PARP1 (0.40) PARP1ALDH1A1HSD11B1
SCHEMBL4053934 0.72 HSD11B1 (0.53) PARP1ALDH1A1MEN1KMT2AHSD11B1
SCHEMBL17633174 0.71 F11 (0.44) ALDH1A1TMPRSS4
SCHEMBL29076911 0.70 F11 (0.39) PARP1JAK2ALDH1A1MEN1KMT2A
SCHEMBL30561093 0.70 F11 (0.39) PARP1JAK2ALDH1A1MEN1KMT2A
SCHEMBL29417027 0.69 PARP1 (0.44) PARP1ALDH1A1PTGESHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015116885-A1 MACROCYCLES WITH AROMATIC P2' GROUPS AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-08-06 WO disclosed