SCHEMBL4055281

SCHEMBL4055281

O=Cc1ccsc1CCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 6/20 0.40
DAO P14920 2/20 0.38
CYP2A6 P11509 1/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
BLM P54132 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
FFAR1 O14842 1/20 0.36
GPR52 Q9Y2T5 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10440205 0.88 LTB4R (0.52) LTB4R
SCHEMBL18995061 0.76 CYP2A6 (0.36) CYP2A6MEN1LMNATHRBBLM
SCHEMBL17428932 0.76 CYP2A6 (0.36) CYP2A6MEN1LMNATHRBBLM
SCHEMBL19222446 0.75 CYP2A6 (0.38) CYP2A6MEN1LMNATHRBBLM
SCHEMBL4054148 0.71 LTB4R (0.40) LTB4RDAOKMT2AFFAR1GPR52
SCHEMBL13147505 0.71 LTB4R (0.50) LTB4RDAOFFAR1
SCHEMBL2082912 0.71 HIF1A (0.40) CYP2A6THRBTDP1
SCHEMBL6964424 0.71
SCHEMBL8255788 0.70 TP53 (0.36) DAOMEN1LMNAKMT2ATDP1
SCHEMBL14116384 0.70 DAO (0.37) DAOFFAR1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057162-A2 FUSED HETEROCYCLIC INHIBITORS OF D-AMINO ACID OXIDASE Sepracor Inc. (US) 2009-05-13 EP disclosed
WO-2008005456-A2 FUSED HETEROCYCLIC INHIBITORS OF D-AMINO ACID OXIDASE SEPRACOR INC. (US) 2008-01-10 WO disclosed