SCHEMBL4055412

SCHEMBL4055412

O=S(=O)(c1ccc(C(F)(F)F)cc1)N1CCSc2ccc(-c3ccccc3)cc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.57
NR1H3 Q13133 3/20 0.51
NR1I2 O75469 1/20 0.51
NR1H2 P55055 1/20 0.51
CYP11B1 P15538 1/20 0.48
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
ACLY P53396 1/20 0.41
MCL1 Q07820 1/20 0.41
CCR6 P51684 1/20 0.41
MMP8 P22894 2/20 0.40
KIF11 P52732 2/20 0.40
MMP3 P08254 1/20 0.40
KDM2B Q8NHM5 1/20 0.39
CPT2 P23786 1/20 0.39
CPT1A P50416 1/20 0.39
CPT1B Q92523 1/20 0.39
GBA1 P04062 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1997923 0.88 RORC (0.50) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL1998534 0.85 SCN2A (0.52) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL2001054 0.82 CNR1 (0.57) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL4062546 0.82 RORC (0.53) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL1998946 0.82 PTPN2 (0.52) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL1999370 0.81 CNR1 (0.57) RORCNR1H3NR1I2NR1H2CNR1
SCHEMBL4062540 0.81 RORC (0.52) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL2001224 0.80 NPC1 (0.48) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL1999110 0.79 RORC (0.54) RORCNR1H3NR1I2NR1H2CYP11B1
SCHEMBL2001965 0.78 CA2 (0.46) RORCNR1H3NR1I2NR1H2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009035997-A2 BENZO-FUSED HETEROCYCLES CARA THERAPEUTICS, INC. (US) 2009-03-19 WO disclosed