SCHEMBL4055988

SCHEMBL4055988

N#Cc1ncn(Cc2c(F)cccc2F)c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.41
ADORA1 P30542 1/20 0.41
PKM P14618 1/20 0.39
AXL P30530 2/20 0.35
MERTK Q12866 2/20 0.35
TYRO3 Q06418 1/20 0.35
ROCK2 O75116 1/20 0.34
FLT3 P36888 1/20 0.34
MAPK14 Q16539 1/20 0.34
EED O75530 1/20 0.34
SUZ12 Q15022 1/20 0.34
EZH2 Q15910 1/20 0.34
TSHR P16473 2/20 0.33
MAPK1 P28482 1/20 0.33
CA5A P35218 1/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 1/20 0.33
CUL4A Q13619 1/20 0.32
JAK2 O60674 1/20 0.31
JAK3 P52333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3130833 0.77 ADORA2A (0.47) ADORA2APKMTSHRCYP11B1CYP11B2
SCHEMBL15432504 0.73 CYP11B1 (0.43) ADORA2APKMMAPK14CYP11B1CYP11B2
SCHEMBL4058117 0.71 CDK1 (0.38) PKMJAK2JAK3ALDH1A1
SCHEMBL4063317 0.71 CDK1 (0.34) ADORA2AADORA1PKMCA5AJAK2
SCHEMBL4639433 0.69 SMN1; SMN2 (0.36) PKMROCK2QPCTKDM4EALDH1A1
SCHEMBL14944585 0.69 CYP11B1 (0.40) ADORA1PKMCYP11B1CYP11B2
SCHEMBL21121675 0.68 ALDH1A1 (0.46) ADORA2AADORA1PKMAXLMERTK
SCHEMBL23416501 0.67 ADORA2A (0.60) ADORA2AADORA1AXLMERTKTYRO3
SCHEMBL1301644 0.67 PKM (0.40) ADORA2AADORA1PKMTSHRKDM4E
SCHEMBL23416492 0.67 ADORA2A (0.63) ADORA2AADORA1AXLMERTKTYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034386-A1 DERIVATIVES OF ADENINE AND 8-AZA-ADENINE AND USES THEREOF-796 ASTRAZENECA AB (SE) 2009-03-19 WO disclosed
WO-2009034386-A1 DERIVATIVES OF ADENINE AND 8-AZA-ADENINE AND USES THEREOF-796 ASTRAZENECA AB (SE) 2009-03-19 WO disclosed