SCHEMBL4056355

SCHEMBL4056355

Cc1ncc2[nH]c(=O)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 5/20 0.43
PDE3A Q14432 5/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA13 Q8N1Q1 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
HCAR1 Q9BXC0 9/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30891708 0.78 MAPKAPK2 (0.42) PDE3BPDE3ACA12CA9CA1
SCHEMBL24885835 0.78 TYRO3 (0.49) PDE3BPDE3ACA12CA9CA1
Hydrochloric Acid SCHEMBL30891705 0.76 MAPKAPK2 (0.41) PDE3BPDE3ACA12CA9CA1
SCHEMBL20660448 0.74 HCAR1 (0.41) PDE3BPDE3ACA12CA9CA1
SCHEMBL4535528 0.73 CA12 (0.48) PDE3BPDE3ACA12CA9CA1
SCHEMBL3334033 0.72 PDE3B (0.44) PDE3BPDE3ACA12CA9CA1
SCHEMBL2619211 0.71 BRD4 (0.37) CA1CA4CA6MAPK1
SCHEMBL890167 0.71 NPY5R (0.37) HTT
SCHEMBL4135331 0.70 CA12 (0.46) PDE3BPDE3ACA12CA9HCAR1
SCHEMBL14494403 0.70 CA12 (0.55) PDE3BPDE3ACA12CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009112524-A1 PYRIDOPYRIMIDINES AS PLK1 ( POLO-LIKE KINASE) INHIBITORS 4SC AG (DE) 2009-09-17 WO disclosed