SCHEMBL4058784

SCHEMBL4058784

COc1ccc(C2(C#N)CCc3nc[nH]c(=O)c3C2)c2c3cc(F)ccc3n(C)c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.34
MYLK Q15746 4/20 0.32
SRC P12931 2/20 0.32
EGFR P00533 1/20 0.32
PDPK1 O15530 1/20 0.31
ALDH1A1 P00352 5/20 0.31
HPGD P15428 2/20 0.31
HSD17B10 Q99714 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PARP1 P09874 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
CASP1 P29466 1/20 0.30
HTT P42858 1/20 0.30
CASP7 P55210 1/20 0.30
ATM Q13315 1/20 0.30
PIK3R1 P27986 1/20 0.30
PIK3CA P42336 1/20 0.30
CCNT1 O60563 1/20 0.30
CDK9 P50750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4059762 0.87 TNKS (0.36) KDM4EMYLKALDH1A1HPGDHSD17B10
SCHEMBL4051890 0.86 TNKS (0.35) KDM4EMYLKALDH1A1HPGDHSD17B10
SCHEMBL4053970 0.81 KDM4E (0.31) KDM4EMYLK
SCHEMBL13693820 0.81 PDE4A (0.41) KDM4EMYLKALDH1A1HPGDHSD17B10
SCHEMBL4540659 0.80 KDM4E (0.32) KDM4E
SCHEMBL4061738 0.79 HTR2A (0.31) KDM4EALDH1A1HPGDHSD17B10GLA
SCHEMBL4052813 0.79 KDM4E (0.31) KDM4EALDH1A1HPGDHSD17B10GLA
SCHEMBL13693578 0.79 PIN1 (0.31) KDM4E
SCHEMBL4058008 0.77 PDE4A (0.33) KDM4EMYLKALDH1A1HPGDHSD17B10
SCHEMBL4058781 0.77 MYLK (0.36) MYLKSRCPIK3R1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO claimed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed