SCHEMBL4059082

SCHEMBL4059082

c1ccc(-c2ccon2)c(-c2ccon2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 3/20 0.40
MAPT P10636 1/20 0.40
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRM1 P11229 1/20 0.36
ALDH1A1 P00352 1/20 0.34
PTPRC P08575 1/20 0.32
ALOX15 P16050 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PLCG2 P16885 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29840757 0.84 NPC1 (0.45) MDM2NPC1RAB9AKDM4EMAPT
SCHEMBL5542787 0.84 MDM2 (0.36) MDM2NPC1RAB9AKDM4EMAPT
SCHEMBL29947384 0.84 IDO1 (0.44) MDM2NPC1RAB9AKDM4EMAPT
SCHEMBL2122583 0.84 NPC1 (0.45) MDM2NPC1RAB9AKDM4EMAPT
SCHEMBL29840696 0.84 IDO1 (0.46) NPC1RAB9AKDM4EMAPTCYP1A2
SCHEMBL30538068 0.84 IDO1 (0.44) NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL1176651 0.84 MDM2 (0.36) MDM2NPC1RAB9AKDM4EMAPT
SCHEMBL700662 0.84 ALDH1A1 (0.48) MDM2NPC1RAB9AKDM4EMAPT
SCHEMBL4714608 0.84 CASP3 (0.44) NPC1RAB9AKDM4EMAPTCYP1A2
SCHEMBL2123489 0.84 IDO1 (0.46) NPC1RAB9AKDM4EMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1801107-B1 Process for the preparation of phenylenebisisoxazoles EVONIK DEGUSSA GMBH (DE) 2009-07-15 EP disclosed
EP-1801107-A1 Process for the preparation of phenylenebisisoxazoles Degussa GmbH (DE) 2007-06-27 EP disclosed