SCHEMBL4061100

SCHEMBL4061100

Cc1ccccc1Nc1nc(Cl)nc2c1cnn2C

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.78
HTR2C P28335 1/20 0.65
TP53 P04637 2/20 0.64
PDE2A O00408 7/20 0.61
KDM4E B2RXH2 2/20 0.61
MAPT P10636 2/20 0.61
ALDH1A1 P00352 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
GAA P10253 1/20 0.61
CYP1A2 P05177 2/20 0.57
CYP3A4 P08684 2/20 0.57
CYP2C19 P33261 2/20 0.57
CYP2D6 P10635 1/20 0.57
MEN1 O00255 3/20 0.55
HSD17B10 Q99714 2/20 0.48
HCRTR1 O43613 1/20 0.48
POLB P06746 1/20 0.48
HSP90AA1 P07900 1/20 0.48
CYP2C9 P11712 1/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3950710 0.83 HTR2C (0.63) KMT2AHTR2CTP53KDM4EMAPT
SCHEMBL13943308 0.82 HTR2C (0.76) KMT2AHTR2CTP53KDM4EMAPT
SCHEMBL4057912 0.81 KMT2A (0.64) KMT2AHTR2CTP53KDM4EMAPT
SCHEMBL20558376 0.80 TP53 (0.52) KMT2AHTR2CTP53KDM4EMAPT
SCHEMBL3949781 0.80 HTR2C (0.66) KMT2AHTR2CTP53KDM4EMAPT
SCHEMBL13087256 0.80 GAA (0.78) KMT2AHTR2CPDE2AKDM4EMAPT
SCHEMBL4063948 0.79 KMT2A (0.65) KMT2AHTR2CTP53PDE2AKDM4E
SCHEMBL13943325 0.79 HTR2C (0.65) KMT2AHTR2CTP53
SCHEMBL13943255 0.78 SHMT2 (0.65) KMT2AHTR2CTP53KDM4EMAPT
SCHEMBL22806016 0.78 GAA (0.80) KMT2AHTR2CPDE2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009023978-A1 PYRAZOLO [3,4 -D] PYRIMIDINE COMPOUNDS AND THEIR USE AS MODULATORS OF PROTEIN KINASE ONCALIS AG (CH) 2009-02-26 WO disclosed
EP-2025678-A1 Pyrazolo[3,4-d]pyrimidine compounds and their use as modulators of protein kinase Oncalis AG (CH) 2009-02-18 EP disclosed
EP-2025678-A1 Pyrazolo[3,4-d]pyrimidine compounds and their use as modulators of protein kinase Oncalis AG (CH) 2009-02-18 EP disclosed