SCHEMBL4064005

SCHEMBL4064005

CC(CN(C)C)NC(=O)c1ccc(-c2c(O)[nH]c3ccc([N+](=O)[O-])cc23)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.46
HDAC1 Q13547 1/20 0.46
MAPT P10636 5/20 0.42
ALDH1A1 P00352 5/20 0.42
GAA P10253 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HTT P42858 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
POLB P06746 1/20 0.41
CCNE1 P24864 5/20 0.40
CDK2 P24941 5/20 0.40
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
GSK3A P49840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4062061 0.99 HDAC4 (0.45) HDAC4HDAC1MAPTALDH1A1GAA
SCHEMBL4065919 0.80 MAPT (0.51) MAPTALDH1A1MEN1KMT2APOLB
SCHEMBL4065913 0.80 MAPT (0.51) MAPTALDH1A1MEN1KMT2APOLB
Hydrochloric Acid SCHEMBL27601566 0.78 CCNE1 (0.39) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL4060329 0.78 CCNE1 (0.46) MAPTALDH1A1GAAKDM4EMEN1
SCHEMBL4234383 0.76 PARP1 (0.47) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL4057858 0.74 TLR9 (0.42) CCNE1CDK2CDK5CDK5R1GSK3A
Hydrochloric Acid SCHEMBL4065193 0.74 FLT3 (0.39) MEN1KMT2ACCNE1CDK2CDK5
Hydrochloric Acid SCHEMBL3195081 0.74 MAPT (0.49) MAPTALDH1A1GAAKDM4EMEN1
SCHEMBL4061512 0.74 LMNA (0.52) ALDH1A1SMN1; SMN2L3MBTL1CDK2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492785-B9 2-HYDROXY-3-HETEROARYLINDOLE DERIVATIVES AS GSK3 INHIBITORS ASTRAZENECA AB (SE) 2009-10-21 EP claimed
EP-1492785-B1 2-HYDROXY-3-HETEROARYLINDOLE DERIVATIVES AS GSK3 INHIBITORS ASTRAZENECA AB (SE) 2008-12-03 EP claimed