Erythromycin

Erythromycin

SCHEMBL40641

CCCCCCCCCCCCCCCCCC(=O)O.CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@]1(C)O

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Erythromycin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.86
KCNH2 Q12809 5/20 0.86
ABCB1 P08183 2/20 0.86
TSHR P16473 2/20 0.86
LMNA P02545 2/20 0.86
MLNR O43193 2/20 0.86
TDP1 Q9NUW8 1/20 0.86
ALB P02768 1/20 0.86
CNR1 P21554 1/20 0.86
HTR2A P28223 1/20 0.86
AOX1 Q06278 1/20 0.86
CYP1B1 Q16678 1/20 0.86
ABCB11 O95342 2/20 0.82
ABCC4 O15439 1/20 0.82
SLCO1B3 Q9NPD5 3/20 0.80
SLCO1B1 Q9Y6L6 3/20 0.80
MAPK1 P28482 2/20 0.80
AR P10275 1/20 0.80
PGR P06401 1/20 0.75
HTR1A P08908 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Erythromycin SCHEMBL11340609 1.00 CYP3A4 (0.86) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL11340606 1.00 CYP3A4 (0.86) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL536998 1.00 CYP3A4 (0.86) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL29116300 1.00 CYP3A4 (0.86) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL10899622 0.99 CYP3A4 (0.84) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL10899617 0.99 CYP3A4 (0.84) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL7056963 0.95 CYP3A4 (0.93) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL7056958 0.95 CYP3A4 (0.93) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL10897935 0.94 CYP3A4 (0.83) CYP3A4KCNH2ABCB1TSHRLMNA
Erythromycin SCHEMBL9487690 0.94 CYP3A4 (0.94) CYP3A4KCNH2ABCB1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5071 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250228841-A1 COMPOSITIONS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES APTORUM THERAPEUTICS LTD (HK) 2025-07-17 US claimed
US-12285471-B2 Methods for treating pulmonary disease using inter-alpha inhibitor proteins PROTHERA BIOLOGICS, INC. (US) 2025-04-29 US claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
US-20250099557-A1 ANTIBIOTIC PHARMACEUTICAL COMPOSITION CAPABLE OF SUBCUTANEOUS ADMINISTRATION SHANGHAI BAO PHARMACEUTICALS CO., LTD. (CN) 2025-03-27 US claimed
CN-119548460-A Erythromycin stearate nano micelle oral liquid preparation and preparation method thereof 神威药业集团有限公司 2025-03-04 CN claimed
CN-118873548-A Anti-liver cancer cell preparation and application thereof 新乡医学院 2024-11-01 CN claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
US-20240173512-A1 METHODS FOR POTENTIATING ANTIMICROBIAL AGENTS STREETERVILLE CAPITAL, LLC 2024-05-30 US claimed
EP-4374848-A1 ANTIBIOTIC PHARMACEUTICAL COMPOSITION CAPABLE OF SUBCUTANEOUS ADMINISTRATION Shanghai Bao Pharmaceuticals Co., Ltd. (CN) 2024-05-29 EP claimed
US-20240122859-A1 EXTENDED RELEASE MULTIPLE UNIT PELLET SYSTEM COMPOSITION AND ITS PROCESS FOR THE PREPARATION NOKHA TRADING LLP (IN) 2024-04-18 US claimed
EP-0277741-A1 Spherical granules having core and their production Takeda Chemical Industries, Ltd. (JP) 1988-08-10 EP claimed
EP-0109102-B1 STORAGE STABLE TOPICAL PHARMACEUTICAL COMPOSITION INCLUDING NITROGEN-CONTAINING STABILIZERS THE PROCTER & GAMBLE COMPANY (US) 1988-01-20 EP claimed
EP-0109102-A2 Storage stable topical pharmaceutical composition including nitrogen-containing stabilizers THE PROCTER & GAMBLE COMPANY (US) 1984-05-23 EP claimed
EP-0027286-B1 ANTI-ACNE COMPOSITION COMPRISING DIISOPROPYL SEBACATE THE PROCTER & GAMBLE COMPANY (US) 1984-02-08 EP claimed
US-4369172-A Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose FOREST LABORATORIES INC. (US) 1983-01-18 US claimed
US-4299826-A TOPICAL APPLICATION OF ERYTHROMYCIN OR DERIVATIVES THE PROCTER & GAMBLE COMPANY (US) 1981-11-10 US claimed
EP-0001871-B1 AN ERYTHROMYCIN COMPOUND, A PROCESS FOR PREPARING THE COMPOUND AND COMPOSITIONS CONTAINING THE COMPOUND USEFUL IN THE TREATMENT OF ACNE THE PROCTER & GAMBLE COMPANY (US) 1981-07-29 EP claimed
EP-0027286-A2 Anti-acne composition comprising diisopropyl sebacate THE PROCTER & GAMBLE COMPANY (US) 1981-04-22 EP claimed
US-4261982-A ZINC ERYTHROMYCIN FOR ACNE THE PROCTER & GAMBLE COMPANY (US) 1981-04-14 US claimed
EP-0001871-A1 An erythromycin compound, a process for preparing the compound and compositions containing the compound useful in the treatment of acne THE PROCTER & GAMBLE COMPANY (US) 1979-05-16 EP claimed