SCHEMBL4064419

SCHEMBL4064419

Cn1ncc(-c2ccc(OCCCCl)cc2)cc1=O.Cn1ncc(-c2ccc(OCCCCl)cc2)cc1=O

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 13/20 0.70
HRH3 Q9Y5N1 5/20 0.49
ADORA2A P29274 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1373281 1.00 HTR3A (0.70) HTR3AHRH3ADORA2ACYP1A2CYP3A4
SCHEMBL1375646 0.82 HTR3A (1.00) HTR3AHRH3KCNH2
SCHEMBL1372915 0.82 HTR3A (1.00) HTR3AHRH3KCNH2
SCHEMBL1373496 0.79 HTR3A (0.56) HTR3A
SCHEMBL1375210 0.78 HTR3A (1.00) HTR3AHRH3KCNH2
SCHEMBL2114693 0.77 HRH3 (0.61) HTR3AHRH3ADORA2ACYP1A2CYP3A4
SCHEMBL3617516 0.76 HTR3A (0.72) HTR3AHRH3CYP1A2CYP2D6CYP19A1
SCHEMBL3610358 0.76 HTR3A (0.71) HTR3AHRH3ADORA2ACYP19A1KCNH2
SCHEMBL4059363 0.75 HTR3A (0.59) HTR3AHRH3KCNH2
SCHEMBL4057349 0.75 HTR3A (0.58) HTR3AHRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069312-A2 PYRIDIZINONE DERIVATIVES Cephalon, Inc. (US) 2009-06-17 EP disclosed
WO-2008013838-A2 PYRIDIZINONE DERIVATIVES CEPHALON, INC. (US) 2008-01-31 WO disclosed