SCHEMBL4066245

SCHEMBL4066245

CC(F)(CCC(CC(O)[CH]Cc1ccccc1OC(F)(F)F)C(=O)NO)C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.40
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PPARG P37231 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
EPHX2 P34913 8/20 0.33
CCR1 P32246 1/20 0.33
SCN9A Q15858 2/20 0.32
ALOX5 P09917 1/20 0.32
NTRK1 P04629 1/20 0.32
GAA P10253 1/20 0.31
F2R P25116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068181 0.87 CCR1 (0.36) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL6832277 0.83 CCR1 (0.41) HDAC3HDAC1HDAC2HDAC6CCR1
SCHEMBL4064274 0.83 CCR1 (0.41) HDAC3HDAC1HDAC2HDAC6CCR1
SCHEMBL4070735 0.83 EPHX1 (0.39) VNN1HDAC1PPARGEPHX2
SCHEMBL4061961 0.81 CYP2D6 (0.40)
SCHEMBL4060776 0.79 CCR1 (0.37) HDAC1HDAC6CCR1
SCHEMBL2675109 0.79 CCR1 (0.38) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL4066473 0.78 CTSC (0.36) CCR1
SCHEMBL4070040 0.77 ANPEP (0.39) VNN1CCR1
SCHEMBL4064283 0.77 TSHR (0.47) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966443-B1 HETEROARYL-HEXANOIC ACID AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS SELECTIVE INHIBITORS OF MIP-1-ALPHA BINDING TO ITS CCR1 RECEPTOR PFIZER (US) 2009-01-28 EP disclosed
US-20020198207-A1 Novel Hexanoic acid derivatives KATH JOHN CHARLES (US) 2002-12-26 US disclosed
US-6403587-B1 AUTOIMMUNE DISEASES, ACUTE AND CHRONIC INFLAMMATORY CONDITIONS, ALLERGIC CONDITIONS, INFECTION ASSOCIATED WITH INFLAMMATION, VIRAL, TRANSPLANTATION TISSUE REJECTION, ATHEROSCLEROSIS, RESTENOSIS, HIV INFECTIVITY, AND PFIZER INC. 2002-06-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020198207-A1 Novel Hexanoic acid derivatives HCAR3, HCAR1, FFAR1 VNN1 3540/4885GRIN1 1536/4885GRIN2B 2149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.