SCHEMBL4066246

SCHEMBL4066246

COc1ccc2nccc(N3C[C@@H]4C[C@H]3CN4CCNC(=O)O)c2n1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.40
CYP8B1 Q9UNU6 1/20 0.39
KCNH2 Q12809 6/20 0.38
SLC2A1 P11166 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4067892 0.83 KCNH2 (0.35) CYP8B1KCNH2
Hydrochloric Acid SCHEMBL5798571 0.83 KCNH2 (0.35) CYP8B1KCNH2
SCHEMBL5905795 0.81 MEN1 (0.37) MAPK1CYP8B1KCNH2
SCHEMBL4063098 0.75 KCNH2 (0.43) KCNH2
SCHEMBL17060472 0.75 PARP1 (0.45) CYP8B1KCNH2
Hydrochloric Acid SCHEMBL4065017 0.75 KCNH2 (0.43) KCNH2
SCHEMBL4070008 0.74 KCNH2 (0.44) CYP8B1KCNH2
SCHEMBL5752149 0.74 CYP8B1 (0.47) CYP8B1KCNH2SLC2A1
SCHEMBL2946390 0.73 KCNH2 (0.40) CYP8B1KCNH2SLC2A1
SCHEMBL1224945 0.71 CHRNB2 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605938-B1 Antibacterial derivatives of napthydrin and quinoline GLAXO GROUP LTD (GB) 2009-02-11 EP disclosed
EP-1605938-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2006-11-22 EP disclosed
EP-1605938-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2005-12-21 EP disclosed
WO-2004087145-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-10-14 WO disclosed