SCHEMBL4067352

SCHEMBL4067352

O=C(Nc1[c]cccc1)Nc1cc(C(F)(F)F)ccc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
KDR P35968 5/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
TSHR P16473 1/20 0.48
PDGFRB P09619 2/20 0.47
TMPRSS4 Q9NRS4 1/20 0.46
RIPK1 Q13546 2/20 0.44
TP53 P04637 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
FLT3 P36888 2/20 0.43
NTRK1 P04629 1/20 0.43
RET P07949 1/20 0.43
LTK P29376 1/20 0.43
CDK8 P49336 1/20 0.43
NTRK3 Q16288 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5271094 0.80 KDR (0.69) CA12CA1CA2CA9KDR
SCHEMBL4798426 0.77 CA12 (0.65) CA12CA1CA2CA9KDR
SCHEMBL6250049 0.77 MEN1 (0.57) MEN1KMT2ATSHRGAAGRIK1
SCHEMBL4797759 0.76 CA12 (0.57) CA12CA1CA2CA9KDR
SCHEMBL9725165 0.75 SMN1; SMN2 (0.44) CA12CA1CA2CA9MEN1
SCHEMBL171921 0.75 CA12 (0.58) CA12CA1CA2CA9KDR
SCHEMBL60290 0.74 KIF11 (0.63) CA12CA1CA2CA9KDR
SCHEMBL29572624 0.74 KIF11 (0.63) CA12CA1CA2CA9KDR
SCHEMBL21750985 0.73 MEN1 (0.59) CA12CA1CA2CA9KDR
SCHEMBL21750852 0.73 CA12 (0.70) CA12CA1CA2CA9KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877409-B1 SUBSTITUTED PYRROLO-PYRIDINES, COMPOSITION CONTAINING THEM, METHOD FOR THEIR PRODUCING AND USE THEREOF AVENTIS PHARMA SA (FR) 2009-06-17 EP claimed