SCHEMBL4067505

SCHEMBL4067505

Cc1nc2c(O[C@@H]3SC[C@@H](O)[C@H](O)[C@H]3O)cccn2c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2D6 P10635 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 2/20 0.44
ATP4A P20648 5/20 0.36
ATP4B P51164 5/20 0.36
PDE10A Q9Y233 2/20 0.32
GUCY1B2 O75343 4/20 0.32
GUCY1A2 P33402 4/20 0.32
GUCY1A1 Q02108 4/20 0.32
GUCY1B1 Q02153 4/20 0.32
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
MEN1 O00255 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4067513 1.00 CYP1A2 (0.44) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4066590 0.81 ADORA3 (0.35)
SCHEMBL4066596 0.81 ADORA3 (0.35)
SCHEMBL4066336 0.79 PSEN1 (0.32) PDE10APSEN1PSEN2APH1BNCSTN
SCHEMBL4066331 0.79 PSEN1 (0.32) PDE10APSEN1PSEN2APH1BNCSTN
SCHEMBL4066131 0.76 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4066126 0.76 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4066428 0.75 SSTR4 (0.36)
SCHEMBL4066424 0.75 SSTR4 (0.36)
SCHEMBL4062013 0.74 HTR4 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041153-B1 NEW 5-THIOXYLOPYRANOSE DERIVATIVES FOURNIER LAB SA (FR) 2009-10-21 EP disclosed