SCHEMBL4068504

SCHEMBL4068504

CCOC(=O)Oc1cnc(Nc2ccccn2)nc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.46
GRM5 P41594 4/20 0.41
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
NPC1 O15118 2/20 0.40
CCND3 P30281 2/20 0.40
CCNK O75909 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CDK9 P50750 1/20 0.40
CDK6 Q00534 1/20 0.40
NOS2 P35228 1/20 0.40
RAB9A P51151 1/20 0.40
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
JAK2 O60674 2/20 0.39
JAK1 P23458 2/20 0.39
TYK2 P29597 2/20 0.39
JAK3 P52333 2/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4071889 0.82 NPC1 (0.57) NPC1RAB9AGAAMAPTALDH1A1
SCHEMBL3649101 0.77 RXFP1 (0.50) GRM5NPC1NOS2RAB9AGAA
SCHEMBL4070689 0.77 CDK4 (0.55) CDK5CDK5R1CCND3CCNKCCNA2
SCHEMBL10584431 0.74 ALDH1A1 (0.42) NPC1RAB9AMAPTHTTMEN1
SCHEMBL4065020 0.69 CCND3 (0.43) GRM5CDK5CDK5R1CCND3CCNK
SCHEMBL30923288 0.69 JAK3 (0.49) GRM5CCND3CCNKCCNA2CDK2
SCHEMBL4065994 0.69 CCNA2 (0.45) PTK2GRM5CDK5CDK5R1NPC1
SCHEMBL8516383 0.68 TSHR (0.52) MAPTMEN1ALDH1A1KMT2AKDM4E
SCHEMBL16694984 0.68 MAPT (0.43) GRM5CCNA2CDK2MAPTHTT
SCHEMBL4069536 0.67 CDK4 (0.54) CCND3CCNKCCNA2CDK2CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1590341-B1 2-AMINOPYRIDINE SUBSTITUTED HETEROCYCLES AS INHIBITORS OF CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2009-06-17 EP claimed