SCHEMBL4068804

SCHEMBL4068804

CCCCc1nc2c(C)nc3ccc(O)cc3c2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
GPR84 Q9NQS5 5/20 0.37
GSK3B P49841 1/20 0.36
TYR P14679 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
ESRRB O95718 1/20 0.36
ESR1 P03372 1/20 0.36
ESRRA P11474 1/20 0.36
ESR2 Q92731 1/20 0.36
PSMB5 P28074 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16694954 0.80 MEN1 (0.44) PARP1KMT2A
SCHEMBL26628009 0.78 KDM4E (0.48) PARP1ALDH1A1KMT2AGAA
SCHEMBL13111952 0.76 PARP1 (0.66) PARP1GPR84GSK3BESRRBESR1
SCHEMBL21815012 0.73 KMT2A (0.58) KMT2AGAAPKMTSHR
SCHEMBL4063897 0.72 ALOX5 (0.34) ALDH1A1KMT2AGAAPKMTSHR
SCHEMBL2270614 0.69 GPR84 (0.43) GPR84
SCHEMBL9038851 0.68 PARP1 (0.57) PARP1TLR7
SCHEMBL6653127 0.67 PARP1 (0.46) PARP1GPR84KMT2A
SCHEMBL30634373 0.66 TLR7 (0.46) TLR7
SCHEMBL22445008 0.66 CETP (0.41) PARP1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658076-A4 ARYLOXY AND ARYLALKYLENEOXY SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES CO (US) 2009-02-25 EP disclosed
EP-1658076-A1 ARYLOXY AND ARYLALKYLENEOXY SUBSTITUTED IMIDAZOQUINOLINES 3M Innovative Properties Company (US) 2006-05-24 EP disclosed
WO-2005020999-A1 ARYLOXY AND ARYLALKYLENEOXY SUBSTITUTED IMIDAZOQUINOLINES 3M INNOVATIVE PROPERTIES COMPANY (US) 2005-03-10 WO disclosed