SCHEMBL4069047

SCHEMBL4069047

FC(F)(F)c1cccc(N2CC[CH]CC2)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.68
SIGMAR1 Q99720 3/20 0.68
HTR3E A5X5Y0 1/20 0.68
HTR3B O95264 1/20 0.68
HTR1D P28221 1/20 0.68
HTR2C P28335 1/20 0.68
HTR3A P46098 1/20 0.68
HTR3D Q70Z44 1/20 0.68
HTR3C Q8WXA8 1/20 0.68
MAPT P10636 3/20 0.66
THRB P10828 1/20 0.66
TSHR P16473 4/20 0.54
LMNA P02545 4/20 0.54
NPSR1 Q6W5P4 3/20 0.54
HTT P42858 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
POLB P06746 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4076837 0.90 ALDH1A1 (0.59) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL28226906 0.89 ALDH1A1 (0.77) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL12706910 0.85 ALDH1A1 (0.72) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL6257153 0.84 ALDH1A1 (0.70) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL4154584 0.83 ALDH1A1 (0.59) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
Hydrochloric Acid SCHEMBL10515108 0.82 MAPT (0.71) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL11874981 0.81 ALDH1A1 (0.68) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL1101976 0.81 ALDH1A1 (0.74) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL220303 0.81 ALDH1A1 (0.66) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL7295918 0.81 ALDH1A1 (0.66) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1415986-B1 SPIRO ISOBENZOFURANES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS BANYU PHARMA CO LTD (JP) 2009-04-08 EP disclosed
US-7205417-B2 Spiro compounds BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-04-17 US disclosed