SCHEMBL4069350

SCHEMBL4069350

CC(C)S(=O)(=O)Nc1ccc2c(c1)S(=O)(=O)C=C(c1c(O)c3cc(F)ccc3n(Cc3ccc(F)cc3)c1=O)N2

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.38
NR1I2 O75469 1/20 0.38
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
PARG Q86W56 6/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC8 Q9BY41 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
BRPF1 P55201 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3929676 0.92 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4068112 0.91 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL3920862 0.90 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4075666 0.89 CYP2C9 (0.37) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4068258 0.87 CYP2C9 (0.37) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4073002 0.87 CYP2C9 (0.42) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL3922950 0.87 CYP2C9 (0.40) CYP2C9NR1I2HDAC1HDAC6HDAC8
SCHEMBL4066606 0.87 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL3922961 0.86 ERCC5 (0.36) CYP2C9NR1I2PARGPTGDR2MAPT
SCHEMBL3930411 0.86 PTGDR2 (0.36) CYP2C9NR1I2PTGS1PTGS2PARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2009-07-29 EP claimed