SCHEMBL4073002

SCHEMBL4073002

O=c1c(C2=CS(=O)(=O)c3cc(NS(=O)(=O)C4CC4)ccc3N2)c(O)c2cc(F)ccc2n1Cc1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.42
NR1I2 O75469 1/20 0.42
MAP2K4 P45985 2/20 0.35
PARG Q86W56 2/20 0.34
HDAC1 Q13547 7/20 0.34
HDAC6 Q9UBN7 7/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC4 P56524 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC9 Q9UKV0 2/20 0.33
HDAC5 Q9UQL6 2/20 0.33
MAP2K7 O14733 1/20 0.33
EPHX2 P34913 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
KIT P10721 1/20 0.33
BRD4 O60885 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065684 0.90 CYP2C9 (0.54) CYP2C9NR1I2MAP2K4PARGMAP2K7
SCHEMBL3920862 0.89 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL3929676 0.89 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4068112 0.89 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4066606 0.87 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4069350 0.87 CYP2C9 (0.38) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL4075666 0.87 CYP2C9 (0.37) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL3922950 0.86 CYP2C9 (0.40) CYP2C9NR1I2HDAC1HDAC6HDAC8
SCHEMBL3930411 0.86 PTGDR2 (0.36) CYP2C9NR1I2PARGPTGDR2
SCHEMBL4068258 0.85 CYP2C9 (0.37) CYP2C9NR1I2PARGHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2009-07-29 EP claimed