SCHEMBL4075666

SCHEMBL4075666

CCCS(=O)(=O)Nc1ccc2c(c1)S(=O)(=O)C=C(c1c(O)c3cc(F)ccc3n(Cc3ccc(F)cc3)c1=O)N2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.37
NR1I2 O75469 1/20 0.37
PARG Q86W56 5/20 0.34
PTGDR2 Q9Y5Y4 3/20 0.34
BRD4 O60885 2/20 0.34
HDAC1 Q13547 4/20 0.34
HDAC6 Q9UBN7 4/20 0.34
HDAC8 Q9BY41 2/20 0.34
KIT P10721 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
NR3C1 P04150 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068258 0.96 CYP2C9 (0.37) CYP2C9NR1I2PARGPTGDR2BRD4
SCHEMBL4068112 0.95 CYP2C9 (0.39) CYP2C9NR1I2PARGPTGDR2BRD4
SCHEMBL3929676 0.91 CYP2C9 (0.39) CYP2C9NR1I2PARGPTGDR2BRD4
SCHEMBL3920862 0.89 CYP2C9 (0.39) CYP2C9NR1I2PARGPTGDR2HDAC1
SCHEMBL3922950 0.89 CYP2C9 (0.40) CYP2C9NR1I2PTGDR2BRD4HDAC1
SCHEMBL4069350 0.89 CYP2C9 (0.38) CYP2C9NR1I2PARGPTGDR2HDAC1
SCHEMBL4072462 0.88 CYP2C9 (0.52) CYP2C9NR1I2PARGPTGDR2BRD4
SCHEMBL4073002 0.87 CYP2C9 (0.42) CYP2C9NR1I2PARGPTGDR2BRD4
SCHEMBL4066606 0.86 CYP2C9 (0.39) CYP2C9NR1I2PARGHDAC1HDAC6
SCHEMBL3922961 0.86 ERCC5 (0.36) CYP2C9NR1I2PARGPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2009-07-29 EP claimed