SCHEMBL4069505

SCHEMBL4069505

NC(=O)C1CC(F)(F)CC[C@]1(O)[C@H](C[C@@H](O)[CH]Cc1ccccc1)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.36
LTB4R Q15722 2/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
LTB4R2 Q9NPC1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7581422 1.00 CCR1 (0.36) CCR1LTB4RCHRM2CHRM1CHRM3
SCHEMBL4063721 0.84 LTB4R (0.36) CCR1LTB4RLTB4R2
SCHEMBL4065572 0.83 CCR1 (0.34) CCR1LTB4RLTB4R2
SCHEMBL6836075 0.83 CCR1 (0.34) CCR1LTB4RLTB4R2
SCHEMBL4059663 0.82 CCR1 (0.35) CCR1LTB4RLTB4R2
SCHEMBL4066914 0.80 MMP1 (0.33)
SCHEMBL2676480 0.79 CCR1 (0.38) CCR1
SCHEMBL4060331 0.78 CCR1 (0.35) CCR1LTB4RLTB4R2
SCHEMBL4065712 0.77 SMN1; SMN2 (0.37) CCR1LTB4RLTB4R2
SCHEMBL7581837 0.77 SMN1; SMN2 (0.37) CCR1LTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966443-B1 HETEROARYL-HEXANOIC ACID AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS SELECTIVE INHIBITORS OF MIP-1-ALPHA BINDING TO ITS CCR1 RECEPTOR PFIZER (US) 2009-01-28 EP disclosed