SCHEMBL4069830

SCHEMBL4069830

O=C(O)c1cc(Cl)c(Cl)c(O)c1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
TSHR P16473 3/20 0.50
CDK2 P24941 2/20 0.48
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2B Q13224 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
PKM P14618 2/20 0.43
AKR1C4 P17516 1/20 0.42
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28740310 0.86 CDK2 (0.48) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL8065086 0.86 TSHR (0.59) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL29186007 0.83 ALDH1A1 (0.55) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL1354508 0.81 PKM (0.50) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL30752461 0.79 TSHR (0.55) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL29185998 0.79 TSHR (0.55) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL27461738 0.79 DPP4 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL29186004 0.78 AKR1C2 (0.44) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL29186005 0.77 ALDH1A1 (0.46) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL11030713 0.76 ALDH1A1 (0.55) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737831-A4 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LTD (AU) 2009-07-22 EP disclosed
EP-1737831-A1 NEUROLOGICALLY-ACTIVE COMPOUNDS Prana Biotechnology Limited (AU) 2007-01-03 EP disclosed
WO-2005095360-A1 NEUROLOGICALLY-ACTIVE COMPOUNDS PRANA BIOTECHNOLOGY LIMITED (AU) 2005-10-13 WO disclosed