SCHEMBL4070711

SCHEMBL4070711

CC1(c2cccc(O)c2)C=C(c2cc(Cl)ccc2F)CN1C(=O)NC1CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.42
KIF11 P52732 8/20 0.41
CHRM1 P11229 3/20 0.38
CHRM3 P20309 3/20 0.38
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
HTR4 Q13639 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
ADAM17 P78536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4062105 0.77 KIF11 (0.59) KCNH2KIF11CHRM1CHRM3CHRM2
SCHEMBL27607778 0.76 KIF11 (0.47) KCNH2KIF11
SCHEMBL4066735 0.76 KIF11 (0.47) KCNH2KIF11
SCHEMBL4070705 0.73 KIF11 (0.44) KCNH2KIF11CHRM1CHRM3CHRM2
SCHEMBL27607773 0.71 KCNH2 (0.46) KCNH2KIF11
SCHEMBL4061574 0.71 KCNH2 (0.46) KCNH2KIF11
SCHEMBL4058060 0.69 KIF11 (0.56) KCNH2KIF11
SCHEMBL4067160 0.68 KIF11 (0.54) KCNH2KIF11
SCHEMBL4058859 0.66 KIF11 (0.87) KCNH2KIF11
SCHEMBL4246685 0.64 KIF11 (0.47) KCNH2KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515724-B1 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2009-10-21 EP claimed