SCHEMBL4071801

SCHEMBL4071801

CCCCN(c1nc2ccccc2n1CC)c1nc2c(Br)c(Br)ccc2n1CC.[Ni]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.39
HTT P42858 2/20 0.39
CYP2D6 P10635 1/20 0.39
TLR8 Q9NR97 3/20 0.38
NPSR1 Q6W5P4 3/20 0.37
LMNA P02545 2/20 0.37
PKM P14618 1/20 0.37
GLA P06280 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL228862 0.82 CYP1A2 (0.47) CYP1A2HTTCYP2D6TLR8NPSR1
SCHEMBL12930508 0.66 HTT (0.57) CYP1A2HTTCYP2D6NPSR1LMNA
SCHEMBL230441 0.64 HTT (0.62) CYP1A2HTTCYP2D6NPSR1LMNA
SCHEMBL9697100 0.61 HTT (0.48) CYP1A2HTTCYP2D6NPSR1LMNA
SCHEMBL6142135 0.61 MEN1 (0.66) TLR8LMNAPKMGLAKDM4E
SCHEMBL230641 0.60 ALDH1A1 (0.70) CYP1A2HTTCYP2D6NPSR1LMNA
SCHEMBL10325213 0.60 MEN1 (0.64) TLR8LMNAPKMGLAKDM4E
SCHEMBL19529567 0.60 TLR8 (0.48) CYP1A2HTTCYP2D6TLR8NPSR1
SCHEMBL230862 0.60 ALDH1A1 (0.51) CYP1A2HTTCYP2D6NPSR1LMNA
SCHEMBL981293 0.59 KDM4E (0.67) CYP1A2HTTCYP2D6NPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2082005-A1 LIGAND EXCHANGE THERMOCHROMIC, (LETC), SYSTEMS Pleotint, L.L.C. (US) 2009-07-29 EP disclosed
WO-2008028128-A1 LIGAND EXCHANGE THERMOCHROMIC, (LETC), SYSTEMS PLEOTINT, L.L.C. (US) 2008-03-06 WO disclosed